Rational design of VHL-recruiting KRASG12C proteolysis-targeting chimeras based on molecular dynamics simulation

Shiyang Sun, Ning Yang, Yaqiu Mao, Ting Wei, Pengli Wei, Tingting Yang, Yixin Zhang, Jian Yan, Changkai Jia, Yi Li, Xu Cai, Zhiyuan Zhao, Xuesong Feng, Xiaomei Zhuang, Wenpeng Zhang, Junhai Xiao, Pengyun Li, Zhibing Zheng, Song Li

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Chinese Chemical Letters ›› 2026, Vol. 37 ›› Issue (02) : 110992. DOI: 10.1016/j.cclet.2025.110992
Communications

Rational design of VHL-recruiting KRASG12C proteolysis-targeting chimeras based on molecular dynamics simulation

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